040-000-527 Azilsartan Medoxomil

SKU: 040-000-527 Category:
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Type Active Pharmaceutical ingredient
CAS No. 863031-21-4
Chemical Formula C30H24N4O8
Appearance white powder
Packaging 100mg, 500mg, 1g, 5g
Assay ≥98%
Related Products Valsartan, Irbesartan, Olmesartan Medoxomil
Description

Description

Azilsartan Medoxomil Introduction

Azilsartan Medoxomil is a prodrug that is rapidly converted to the active moiety, azilsartan (TAK-536), by ester hydrolysis in the gut and plasma. In vascular smooth muscle and adrenal glands, Azilsartan selectively blocks the binding of angiotensin II to the AT1 (angiotensin II type 1) receptor, thereby promoting vasodilation and reducing the effects of aldosterone. It is a potent angiotensin II type 1 (AT1) receptor antagonist that inhibits RAAS with >10,000-fold selectivity over AT2 for the treatment of hypertension.

Azilsartan Medoxomil Specification

Appearance white powder
Melting Point 160-161℃
Density 1.45
Content 98.0%
Storage Condition 2-8℃
Packaging 100mg, 500mg, 1g, 5g

 

Azilsartan Medoxomil Applications

Azilsartan Medoxomil is a prodrug that is rapidly converted to the active moiety, azilsartan (TAK-536), by ester hydrolysis in the gut and plasma.